SCHEMBL4030776

SCHEMBL4030776

CNC(=O)CC(N[S+]([O-])C(C)(C)C)c1ccc(F)cn1

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
APLNR P35414 1/20 0.34
NR1I2 O75469 1/20 0.32
NTRK1 P04629 1/20 0.31
CNR1 P21554 1/20 0.31
CNR2 P34972 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4023097 0.88 APLNR (0.35) APLNRNR1I2CNR1CNR2
SCHEMBL4196483 0.83 CXCR1 (0.35) APLNRNR1I2NTRK1
SCHEMBL3946528 0.81 APLNR (0.34) APLNRNTRK1CNR1CNR2
SCHEMBL4184543 0.79 APLNR (0.38) APLNRNTRK1
SCHEMBL4021434 0.77 HDAC6 (0.32) APLNR
SCHEMBL4019567 0.74 HDAC6 (0.30)
SCHEMBL1439307 0.74 HDAC6 (0.30)
SCHEMBL1693207 0.74 HDAC6 (0.30)
SCHEMBL3015031 0.74 HDAC6 (0.30)
SCHEMBL3238364 0.74 HDAC6 (0.41) APLNRNR1I2NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009095712-A2 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2009-08-06 WO disclosed
WO-2009016410-A2 CHEMICAL COMPOUNDS 831 ASTRAZENECA AB (SE) 2009-02-05 WO disclosed