SCHEMBL4196483

SCHEMBL4196483

CCOC(=O)CC(N[S+]([O-])C(C)(C)C)c1ccc(F)cn1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR1 P25024 1/20 0.35
CXCR2 P25025 1/20 0.35
POLB P06746 2/20 0.34
APLNR P35414 1/20 0.32
NR1I2 O75469 1/20 0.32
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
P2RX3 P56373 1/20 0.32
CYP1A2 P05177 2/20 0.32
MAPT P10636 6/20 0.32
LMNA P02545 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
TP53 P04637 1/20 0.32
MAOB P27338 1/20 0.31
NTRK1 P04629 1/20 0.31
BACE1 P56817 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4023097 0.85 APLNR (0.35) APLNRNR1I2
SCHEMBL4030776 0.83 APLNR (0.34) APLNRNR1I2NTRK1
SCHEMBL18640937 0.82 SMN1; SMN2 (0.44) MEN1KMT2ACYP1A2LMNACYP2C19
SCHEMBL31362647 0.82 SMN1; SMN2 (0.44) MEN1KMT2ACYP1A2LMNACYP2C19
SCHEMBL25235485 0.80 KCNB1 (0.34) CYP1A2MAPTLMNACYP2C9CYP2C19
SCHEMBL20142638 0.79 ALDH1A1 (0.46) POLBMEN1KMT2ACYP1A2MAPT
SCHEMBL18361518 0.78 THRB (0.34) POLBMEN1KMT2ACYP1A2MAPT
SCHEMBL18361519 0.78 THRB (0.34) POLBMEN1KMT2ACYP1A2MAPT
SCHEMBL3946528 0.78 APLNR (0.34) APLNRNTRK1
SCHEMBL13437542 0.77 BACE1 (0.33) POLBAPLNRMEN1KMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009016410-A2 CHEMICAL COMPOUNDS 831 ASTRAZENECA AB (SE) 2009-02-05 WO disclosed