SCHEMBL4032463

SCHEMBL4032463

COc1ccc(NC(=O)ON2CCC3(CC2)NC(Cc2ccccc2)C(=O)N3Cc2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CCR3 P51677 2/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
LMNA P02545 2/20 0.43
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
ACHE P22303 1/20 0.41
BACE1 P56817 1/20 0.41
MAPT P10636 2/20 0.41
GLA P06280 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
FAAH O00519 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CHRM3 P20309 1/20 0.40
GAA P10253 1/20 0.40
HTT P42858 1/20 0.40
BCHE P06276 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4035453 0.92 BCHE (0.47) CCR3MEN1KMT2ALMNAACHE
SCHEMBL4040634 0.79 BCHE (0.44) CCR3KMT2AACHEFAAHALDH1A1
SCHEMBL1801528 0.78 CXCR3 (0.57) MEN1KMT2ACYP2D6SIGMAR1ALDH1A1
SCHEMBL4039209 0.78 CXCR3 (0.38) KMT2AL3MBTL1
SCHEMBL2940834 0.78 CXCR3 (0.38) KMT2AL3MBTL1
SCHEMBL1801540 0.78 CYP2D6 (0.41) MEN1KMT2ASMN1; SMN2LMNACYP2D6
SCHEMBL2940899 0.78 CYP2D6 (0.41) MEN1KMT2ASMN1; SMN2LMNACYP2D6
SCHEMBL2940902 0.78 CYP2D6 (0.41) MEN1KMT2ASMN1; SMN2LMNACYP2D6
SCHEMBL3914967 0.78 FAAH (0.52) CYP2D6CYP2C19MAPTFAAHALDH1A1
SCHEMBL2933989 0.78 CYP2D6 (0.54) MEN1KMT2ASMN1; SMN2CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP claimed
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP disclosed