SCHEMBL4035453

SCHEMBL4035453

O=C(Nc1ccccc1)ON1CCC2(CC1)NC(Cc1ccccc1)C(=O)N2Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BCHE P06276 7/20 0.47
ACHE P22303 6/20 0.45
MAOB P27338 3/20 0.45
GAA P10253 2/20 0.41
PKM P14618 1/20 0.41
KMT2A Q03164 2/20 0.40
DRD2 P14416 1/20 0.40
DRD4 P21917 1/20 0.40
DRD3 P35462 1/20 0.40
FAAH O00519 1/20 0.39
CCR3 P51677 1/20 0.39
ALDH1A1 P00352 1/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4032463 0.92 CCR3 (0.47) BCHEACHEGAAKMT2AFAAH
SCHEMBL4040634 0.86 BCHE (0.44) BCHEACHEMAOBGAAPKM
SCHEMBL3914967 0.85 FAAH (0.52) GAAPKMFAAHALDH1A1MAPT
SCHEMBL3914881 0.82 KMT2A (0.51) KMT2AALDH1A1MEN1LMNAMAPT
SCHEMBL2940834 0.82 CXCR3 (0.38) KMT2A
SCHEMBL4039209 0.82 CXCR3 (0.38) KMT2A
SCHEMBL3926088 0.80 CXCR3 (0.41) GAA
SCHEMBL1797763 0.78 CYP2D6 (0.51) GAAKMT2AALDH1A1MEN1
SCHEMBL4032741 0.78 ATM (0.44) KMT2ACCR3ALDH1A1MEN1MAPT
Hydrochloric Acid SCHEMBL1800654 0.77 CYP2D6 (0.50) GAAKMT2AALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP claimed
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP disclosed