SCHEMBL4040634

SCHEMBL4040634

O=C(Nc1ccccc1)OSN1CCC2(CC1)NC(Cc1ccccc1)C(=O)N2Cc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BCHE P06276 6/20 0.44
MAOB P27338 3/20 0.41
ACHE P22303 2/20 0.41
PKM P14618 2/20 0.40
GAA P10253 1/20 0.40
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
DRD3 P35462 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 1/20 0.36
FAAH O00519 1/20 0.35
CCR3 P51677 1/20 0.35
CXCR3 P49682 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4035453 0.86 BCHE (0.47) BCHEMAOBACHEPKMGAA
SCHEMBL4032241 0.86 KMT2A (0.41) GAAKMT2AALDH1A1CCR3
SCHEMBL4035232 0.84 FAAH (0.39) DRD2DRD4DRD3ALDH1A1FAAH
SCHEMBL3914967 0.82 FAAH (0.52) PKMGAAALDH1A1FAAH
SCHEMBL4034900 0.81 CXCR3 (0.40) PKMGAAALDH1A1CXCR3
SCHEMBL3914881 0.80 KMT2A (0.51) KMT2AALDH1A1
SCHEMBL4034612 0.79 ATM (0.40) KMT2AALDH1A1CXCR3
SCHEMBL4032463 0.79 CCR3 (0.47) BCHEACHEGAAKMT2AALDH1A1
SCHEMBL4034807 0.78 CXCR3 (0.39) GAAKMT2AALDH1A1CCR3CXCR3
SCHEMBL3926088 0.78 CXCR3 (0.41) GAACXCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP claimed
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP disclosed
EP-1730144-A1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5|DECAN-2-ONE COMPOUNDS Grünenthal GmbH (DE) 2006-12-13 EP disclosed
WO-2005095398-A1 SUBSTITUTED 1,4,8-TRIAZASPIRO[4.5]DECAN-2-ONE COMPOUNDS Grünenthal GmbH (DE) 2005-10-13 WO disclosed