SCHEMBL4032836

SCHEMBL4032836

Cc1ccnc(CCN(CCCCNC(=O)OC(C)(C)C)Cc2ncccc2C)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 2/20 0.40
DRD2 P14416 3/20 0.38
MAPT P10636 1/20 0.38
ATM Q13315 1/20 0.38
CYP3A4 P08684 2/20 0.38
DYRK1A Q13627 1/20 0.37
TSHR P16473 3/20 0.37
TP53 P04637 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
BRD4 O60885 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
STING1 Q86WV6 1/20 0.36
KDM4E B2RXH2 1/20 0.35
PDPK1 O15530 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4039491 0.88 CYP3A4 (0.44) CXCR4DRD2CYP3A4TSHRL3MBTL1
SCHEMBL4035412 0.87 DRD2 (0.42) CXCR4DRD2CYP3A4TSHRL3MBTL1
SCHEMBL2083428 0.84 CYP3A4 (0.43) CXCR4DRD2CYP3A4DYRK1ATSHR
SCHEMBL4032545 0.82 L3MBTL1 (0.40) CXCR4DRD2CYP3A4TSHRL3MBTL1
SCHEMBL2085707 0.82 CXCR4 (0.64) CXCR4MAPTATMCYP3A4NPSR1
SCHEMBL2085143 0.78 CYP3A4 (0.42) CXCR4MAPTATMCYP3A4DYRK1A
SCHEMBL2086065 0.78 CXCR4 (0.41) CXCR4DRD2CYP3A4DYRK1AL3MBTL1
SCHEMBL4038791 0.77 MAOA (0.45) MAPTATMCYP3A4DYRK1ATSHR
SCHEMBL2083791 0.75 CKS1B (0.41) CXCR4MAPTCYP3A4ALDH1A1NPSR1
SCHEMBL2081783 0.75 BCHE (0.48) CXCR4TP53SMN1; SMN2BRD4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed