SCHEMBL4033159

SCHEMBL4033159

CNC(=O)Oc1[nH]c2cccnc2c1Sc1cccc(F)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 1/20 0.37
TGFBR1 P36897 6/20 0.37
TGFBR2 P37173 5/20 0.37
ALDH1A1 P00352 3/20 0.36
GRM4 Q14833 1/20 0.35
POLB P06746 2/20 0.34
SLC6A9 P48067 1/20 0.34
TUBB4A P04350 1/20 0.34
TUBB P07437 1/20 0.34
TUBA3C P0DPH7 1/20 0.34
TUBA1B P68363 1/20 0.34
TUBA4A P68366 1/20 0.34
TUBB4B P68371 1/20 0.34
TUBB3 Q13509 1/20 0.34
TUBB2A Q13885 1/20 0.34
TUBB8 Q3ZCM7 1/20 0.34
TUBA3E Q6PEY2 1/20 0.34
TUBA1A Q71U36 1/20 0.34
TUBA1C Q9BQE3 1/20 0.34
TUBB6 Q9BUF5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4038485 0.88 TUBB4A (0.40) TYMSTGFBR1TGFBR2ALDH1A1GRM4
SCHEMBL4035517 0.86 TYMS (0.37) TYMSTGFBR1TGFBR2ALDH1A1GRM4
SCHEMBL4042410 0.85 PDE2A (0.42) TGFBR1TGFBR2ALDH1A1TUBB4ATUBB
SCHEMBL2053003 0.76 PTGS2 (0.40) TYMSTGFBR1TGFBR2ALDH1A1GRM4
SCHEMBL4043268 0.76 PKN1 (0.36) TGFBR1TGFBR2GRM4TUBB4ATUBB
SCHEMBL4036370 0.74 PARP1 (0.37) TGFBR1TGFBR2ALDH1A1HPGD
SCHEMBL4036538 0.74 JAK2 (0.48) TGFBR1ALDH1A1GRM4TUBB4ATUBB
SCHEMBL4033058 0.74 TYMS (0.37) TYMSTGFBR1TGFBR2ALDH1A1RAB9A
SCHEMBL4036827 0.74 KDM4E (0.43) TYMSTGFBR1TGFBR2ALDH1A1GRM4
SCHEMBL4033177 0.73 KIF11 (0.42) TGFBR1ALDH1A1GRM4POLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1747220-B1 SUBSTITUTED 1H-PYRROLO[3,2-B, 3,2-C, AND 2,3-C]PYRIDINE-2-CARBOXAMIDES AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE I EPSILON AVENTIS PHARMA INC (US) 2009-04-15 EP claimed