SCHEMBL4035517

SCHEMBL4035517

NC(=O)Oc1[nH]c2cccnc2c1Sc1cccc(F)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 1/20 0.37
RAB9A P51151 2/20 0.35
LMNA P02545 2/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
NPC1 O15118 1/20 0.35
TGFBR1 P36897 2/20 0.35
TGFBR2 P37173 2/20 0.35
GRM4 Q14833 1/20 0.34
RPS6KB1 P23443 1/20 0.34
JAK2 O60674 1/20 0.34
EPHX1 P07099 1/20 0.34
SLC6A9 P48067 1/20 0.33
HAO1 Q9UJM8 1/20 0.33
PIK3CA P42336 1/20 0.33
CDC7 O00311 1/20 0.33
MAPK14 Q16539 1/20 0.33
POLB P06746 1/20 0.32
CA2 P00918 1/20 0.32
CA4 P22748 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4036370 0.88 PARP1 (0.37) ALDH1A1HPGDTGFBR1TGFBR2RPS6KB1
SCHEMBL4036827 0.87 KDM4E (0.43) TYMSRAB9AALDH1A1HPGDNPC1
SCHEMBL4043268 0.87 PKN1 (0.36) RAB9ANPC1TGFBR1TGFBR2GRM4
SCHEMBL4033058 0.87 TYMS (0.37) TYMSRAB9AALDH1A1NPC1TGFBR1
SCHEMBL4033159 0.86 TYMS (0.37) TYMSRAB9ALMNAALDH1A1HPGD
SCHEMBL4033177 0.86 KIF11 (0.42) LMNAALDH1A1TGFBR1GRM4POLB
SCHEMBL4035502 0.86 TUBB4A (0.39) LMNAALDH1A1JAK2
SCHEMBL4036538 0.85 JAK2 (0.48) RAB9ALMNAALDH1A1NPC1TGFBR1
SCHEMBL4035416 0.85 RHEB (0.43) RPS6KB1JAK2MAPK14
SCHEMBL4207716 0.83 MAPT (0.42) RAB9ALMNAALDH1A1HPGDNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1747220-B1 SUBSTITUTED 1H-PYRROLO[3,2-B, 3,2-C, AND 2,3-C]PYRIDINE-2-CARBOXAMIDES AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE I EPSILON AVENTIS PHARMA INC (US) 2009-04-15 EP claimed