SCHEMBL4036370

SCHEMBL4036370

NC(=O)Oc1[nH]c2cccnc2c1Sc1cccc(N)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.37
PLK4 O00444 2/20 0.37
MAP4K4 O95819 2/20 0.37
PIM1 P11309 2/20 0.37
AURKB Q96GD4 2/20 0.37
MKNK2 Q9HBH9 2/20 0.37
STK17A Q9UEE5 2/20 0.37
EGFR P00533 1/20 0.37
ROS1 P08922 1/20 0.37
AXL P30530 1/20 0.37
FLT3 P36888 1/20 0.37
FRK P42685 1/20 0.37
MAP4K2 Q12851 1/20 0.37
NTRK3 Q16288 1/20 0.37
MINK1 Q8N4C8 1/20 0.37
HIPK2 Q9H2X6 1/20 0.37
IRAK4 Q9NWZ3 1/20 0.37
ALK Q9UM73 1/20 0.37
JAK2 O60674 1/20 0.35
PKN1 Q16512 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043268 0.88 PKN1 (0.36) PARP1JAK2PKN1PKN2TGFBR1
SCHEMBL4036827 0.88 KDM4E (0.43) PARP1TGFBR1TGFBR2ALDH1A1KDM4E
SCHEMBL4033058 0.88 TYMS (0.37) JAK2PKN1PKN2TGFBR1TGFBR2
SCHEMBL4035517 0.88 TYMS (0.37) JAK2PKN1PKN2TGFBR1TGFBR2
SCHEMBL4035502 0.87 TUBB4A (0.39) PARP1JAK2PDE5AALDH1A1MEN1
SCHEMBL4036538 0.86 JAK2 (0.48) PARP1JAK2PKN1PKN2TGFBR1
SCHEMBL4034008 0.85 LMNA (0.37) PARP1JAK2PKN1PKN2TGFBR1
SCHEMBL4033177 0.85 KIF11 (0.42) PARP1TGFBR1ALDH1A1KDM4EMEN1
SCHEMBL4207716 0.84 MAPT (0.42) PARP1ALDH1A1KDM4EMEN1HPGD
SCHEMBL4033192 0.84 PKN1 (0.38) PARP1PLK4MAP4K4PIM1AURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1747220-B1 SUBSTITUTED 1H-PYRROLO[3,2-B, 3,2-C, AND 2,3-C]PYRIDINE-2-CARBOXAMIDES AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE I EPSILON AVENTIS PHARMA INC (US) 2009-04-15 EP claimed