SCHEMBL4033737

SCHEMBL4033737

CCC(c1ccc(F)cc1)c1cccnc1C=O

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.37
ALOX12 P18054 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
NFE2L2 Q16236 3/20 0.36
TSHR P16473 2/20 0.35
EPHX2 P34913 1/20 0.34
FAAH O00519 1/20 0.34
NPC1 O15118 1/20 0.33
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.33
ALDH1A1 P00352 2/20 0.33
CYP17A1 P05093 2/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
HPGD P15428 1/20 0.33
CYP19A1 P11511 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5574440 0.88 TSHR (0.43) KDM4ETSHRLMNAPOLBALDH1A1
SCHEMBL21910135 0.77 LMNA (0.45) KDM4EALOX12MEN1KMT2ANPC1
SCHEMBL4035437 0.76 TRPA1 (0.36) KDM4EMEN1KMT2ANFE2L2NPC1
SCHEMBL7089658 0.75 TSHR (0.43) KDM4EMEN1KMT2ATSHRNPC1
SCHEMBL4032446 0.74 NFE2L2 (0.36) NFE2L2POLBALDH1A1
SCHEMBL21911301 0.73 SLC6A2 (0.40) NPC1LMNAPOLBALDH1A1CYP17A1
SCHEMBL23055173 0.73 CYP17A1 (0.38) KDM4EALOX12MEN1KMT2ANFE2L2
SCHEMBL30415398 0.72 TRIM24 (0.32) MEN1KMT2AALDH1A1PKM
SCHEMBL2082260 0.71 GABRA1 (0.39) KDM4EMEN1KMT2ATSHRFAAH
SCHEMBL1179712 0.71 TRIM24 (0.38) KDM4EMEN1KMT2ANFE2L2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed