SCHEMBL4033852

SCHEMBL4033852

O=C(NCc1ccc(F)cc1)C1CN(C(=O)C(c2ccccc2)c2ccccc2)CCN1S(=O)(=O)c1ccc2ncccc2c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.46
NAMPT P43490 1/20 0.44
ALDH1A1 P00352 3/20 0.42
CHRM1 P11229 1/20 0.42
MMP1 P03956 2/20 0.41
MMP3 P08254 2/20 0.41
MMP7 P09237 2/20 0.41
MMP9 P14780 2/20 0.41
FKBP1A P62942 1/20 0.41
ATM Q13315 1/20 0.41
MMP13 P45452 1/20 0.41
LMNA P02545 1/20 0.41
TRPA1 O75762 4/20 0.40
PKM P14618 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4035481 0.90 TSHR (0.49) TSHRNAMPTALDH1A1CHRM1MMP1
SCHEMBL4037487 0.88 MAPT (0.49) TSHRNAMPTALDH1A1LMNAPKM
SCHEMBL4038385 0.86 ALDH1A1 (0.57) ALDH1A1CHRM1PKM
SCHEMBL4042256 0.85 POLB (0.46) ALDH1A1CHRM1MMP1MMP3MMP7
SCHEMBL4042590 0.85 CHRM1 (0.43) NAMPTALDH1A1CHRM1LMNA
SCHEMBL4033849 0.85 MAPK1 (0.53) TSHRALDH1A1LMNA
SCHEMBL4033312 0.85 P2RX7 (0.45)
SCHEMBL4035457 0.84 CHRM5 (0.45) NAMPTCHRM1MMP1MMP3MMP7
SCHEMBL4033365 0.82 SMN1; SMN2 (0.47) ALDH1A1CHRM1MMP1MMP3MMP7
SCHEMBL4034711 0.81 KMT2A (0.41) ALDH1A1CHRM1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1592389-B1 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES SERONO LAB (CH) 2009-04-22 EP claimed