SCHEMBL4035481

SCHEMBL4035481

O=C(NCc1cccnc1)C1CN(C(=O)C(c2ccccc2)c2ccccc2)CCN1S(=O)(=O)c1ccc2ncccc2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.49
KDM4E B2RXH2 1/20 0.49
NAMPT P43490 2/20 0.48
LMNA P02545 2/20 0.46
ALDH1A1 P00352 2/20 0.46
USP2 O75604 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CHRM1 P11229 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
KMT2A Q03164 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MEN1 O00255 1/20 0.43
MAPK1 P28482 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
NPC1 O15118 1/20 0.43
MMP1 P03956 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4033852 0.90 TSHR (0.46) TSHRNAMPTLMNAALDH1A1CHRM1
SCHEMBL4037487 0.86 MAPT (0.49) TSHRKDM4ENAMPTLMNAALDH1A1
SCHEMBL4038385 0.86 ALDH1A1 (0.57) KDM4EALDH1A1USP2CHRM1KMT2A
SCHEMBL4042590 0.85 CHRM1 (0.43) NAMPTLMNAALDH1A1USP2CHRM1
SCHEMBL4042256 0.85 POLB (0.46) LMNAALDH1A1USP2CHRM1MMP1
SCHEMBL4035477 0.85 MAPK1 (0.53) TSHRNAMPTLMNAALDH1A1KMT2A
SCHEMBL4033312 0.85 P2RX7 (0.45) L3MBTL1POLB
SCHEMBL4035457 0.83 CHRM5 (0.45) NAMPTLMNACHRM1MMP1MMP3
SCHEMBL4033365 0.82 SMN1; SMN2 (0.47) LMNAALDH1A1CHRM1KMT2ASMN1; SMN2
SCHEMBL4034711 0.81 KMT2A (0.41) KDM4ELMNAALDH1A1USP2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1592389-B1 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES SERONO LAB (CH) 2009-04-22 EP claimed