SCHEMBL4033953

SCHEMBL4033953

CCCCc1ccc(-c2onc(C)c2N(C(=O)O)C(C)c2ccccc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LPAR1 Q92633 2/20 0.41
TP53 P04637 1/20 0.40
GAA P10253 1/20 0.40
S1PR1 P21453 2/20 0.39
S1PR3 Q99500 1/20 0.39
HSD11B1 P28845 1/20 0.39
LPAR3 Q9UBY5 1/20 0.39
RARB P10826 1/20 0.38
LTB4R2 Q9NPC1 6/20 0.37
DHODH Q02127 1/20 0.37
S1PR4 O95977 1/20 0.37
S1PR5 Q9H228 1/20 0.37
CNR2 P34972 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4034918 0.88 LPAR1 (0.45) LPAR1TP53GAAS1PR1S1PR3
SCHEMBL4028121 0.85 LPAR1 (0.44) LPAR1LPAR3
SCHEMBL4033561 0.83 LPAR1 (0.42) LPAR1LPAR3
SCHEMBL4031584 0.82 LPAR1 (0.43) LPAR1S1PR1LPAR3
SCHEMBL4031919 0.80 TRPA1 (0.50) LPAR1S1PR3LPAR3S1PR4
SCHEMBL4036870 0.79 MAPK1 (0.42) LPAR1LPAR3CNR2
SCHEMBL4030691 0.78 LPAR1 (0.41) LPAR1TP53LPAR3
SCHEMBL4027903 0.78 HTT (0.45) LPAR1TP53GAALPAR3CNR2
SCHEMBL4034953 0.76 LPAR1 (0.52) LPAR1S1PR1S1PR3LPAR3LTB4R2
SCHEMBL4034077 0.76 HDAC3 (0.41) LPAR1LPAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1258484-B1 NOVEL ISOXAZOLE AND THIAZOLE COMPOUNDS AND USE THEREOF AS DRUGS KYOWA HAKKO KIRIN CO LTD (JP) 2009-01-14 EP claimed