SCHEMBL4031919

SCHEMBL4031919

Cc1noc(-c2ccc(C#N)cc2)c1N(C(=O)O)C(C)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.50
EP300 Q09472 6/20 0.40
LPAR1 Q92633 3/20 0.40
LPAR3 Q9UBY5 1/20 0.40
S1PR3 Q99500 2/20 0.38
S1PR4 O95977 1/20 0.38
ALDH1A1 P00352 2/20 0.37
BRD4 O60885 2/20 0.37
ABCC3 O15438 1/20 0.36
ABCC4 O15439 1/20 0.36
ABCB11 O95342 1/20 0.36
CYP2C8 P10632 1/20 0.36
CYP2C9 P11712 1/20 0.36
ABCB4 P21439 1/20 0.36
ABCC2 Q92887 1/20 0.36
SLCO1B3 Q9NPD5 1/20 0.36
SLCO1B1 Q9Y6L6 1/20 0.36
STAT3 P40763 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4028121 0.88 LPAR1 (0.44) TRPA1LPAR1LPAR3ALDH1A1ABCC3
SCHEMBL4036790 0.87 TRPA1 (0.46) TRPA1EP300LPAR1LPAR3ALDH1A1
SCHEMBL4031683 0.85 TRPA1 (0.43) TRPA1EP300LPAR1LPAR3S1PR3
SCHEMBL4033561 0.85 LPAR1 (0.42) TRPA1LPAR1LPAR3ALDH1A1ABCC3
SCHEMBL4031584 0.84 LPAR1 (0.43) TRPA1LPAR1LPAR3ALDH1A1ABCC3
SCHEMBL4036870 0.82 MAPK1 (0.42) LPAR1LPAR3ALDH1A1LMNA
SCHEMBL4030691 0.80 LPAR1 (0.41) LPAR1LPAR3ABCC3ABCC4ABCB11
SCHEMBL4033953 0.80 LPAR1 (0.41) LPAR1LPAR3S1PR3S1PR4
SCHEMBL4027903 0.80 HTT (0.45) LPAR1LPAR3ALDH1A1BRD4STAT3
SCHEMBL4034077 0.78 HDAC3 (0.41) LPAR1LPAR3BRD4STAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1258484-B1 NOVEL ISOXAZOLE AND THIAZOLE COMPOUNDS AND USE THEREOF AS DRUGS KYOWA HAKKO KIRIN CO LTD (JP) 2009-01-14 EP claimed