SCHEMBL4034900

SCHEMBL4034900

O=C(O)SN1CCC2(CC1)NC(Cc1ccccc1)C(=O)N2Cc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 1/20 0.40
CCR5 P51681 5/20 0.39
GAA P10253 3/20 0.38
POLB P06746 1/20 0.38
HDAC1 Q13547 3/20 0.36
HDAC6 Q9UBN7 3/20 0.36
HDAC8 Q9BY41 4/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
PKM P14618 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4038603 0.89 ATM (0.42) CXCR3POLBKDM4EALDH1A1LMNA
SCHEMBL4037470 0.86 GAA (0.44) CXCR3CCR5GAAL3MBTL1KDM4E
SCHEMBL4041207 0.85 PLA2G10 (0.38) CXCR3GAAPOLBHDAC8KDM4E
SCHEMBL3926088 0.85 CXCR3 (0.41) CXCR3CCR5GAAPOLBHDAC1
SCHEMBL1797763 0.83 CYP2D6 (0.51) CXCR3CCR5GAAALDH1A1
SCHEMBL4037625 0.83 ALDH1A1 (0.40) CCR5L3MBTL1KDM4EALDH1A1LMNA
Hydrochloric Acid SCHEMBL1800654 0.82 CYP2D6 (0.50) CXCR3CCR5GAAALDH1A1
SCHEMBL3918198 0.82 GAA (0.41) CXCR3CCR5GAAPOLBHDAC1
SCHEMBL4040634 0.81 BCHE (0.44) CXCR3GAAPKMALDH1A1
SCHEMBL1798600 0.81 NPC1 (0.48) POLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP claimed