SCHEMBL4038579

SCHEMBL4038579

Cc1ncccc1CC(C)c1ccc(Cl)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
FFAR2 O15552 2/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
HRH1 P35367 3/20 0.37
CHRM2 P08172 2/20 0.37
CHRM5 P08912 2/20 0.37
CHRM1 P11229 2/20 0.37
ADRA2B P18089 2/20 0.37
SLC6A2 P23975 2/20 0.37
HRH2 P25021 2/20 0.37
HTR2A P28223 2/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 2/20 0.37
KCNH2 Q12809 2/20 0.37
HRH3 Q9Y5N1 2/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4038116 0.81 L3MBTL1 (0.40) TRPA1MEN1KMT2AFFAR2PTGDR2
SCHEMBL4035579 0.81 TRPA1 (0.42) TRPA1MEN1KMT2AFFAR2PTGDR2
SCHEMBL31256727 0.78 TRPA1 (0.39) TRPA1MEN1KMT2AFFAR2PTGDR2
SCHEMBL4030343 0.76 TRPA1 (0.38) TRPA1MEN1KMT2AFFAR2PTGDR2
SCHEMBL2084548 0.76 GABRA1 (0.47) MEN1KMT2ACYP2C9L3MBTL1FFAR1
SCHEMBL21915781 0.73 C3AR1 (0.37) SLC6A2SLC6A4SLC6A3CYP2C9TSHR
SCHEMBL21401005 0.73 SLC6A2 (0.41) SLC6A2HTR2ASLC6A4SLC6A3HTR2B
SCHEMBL24741410 0.71 P2RX7 (0.37) MEN1KMT2ACYP2C9L3MBTL1FFAR1
SCHEMBL23691145 0.70 C3AR1 (0.37) SLC6A2SLC6A4SLC6A3CYP2D6CYP2C9
SCHEMBL738256 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed