SCHEMBL4035579

SCHEMBL4035579

CC(Cc1cccnc1C=O)c1ccc(Cl)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.42
FFAR2 O15552 5/20 0.42
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
NFE2L2 Q16236 3/20 0.37
P2RX7 Q99572 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
CHRM2 P08172 2/20 0.35
CHRM5 P08912 2/20 0.35
CHRM1 P11229 2/20 0.35
ADRA2B P18089 2/20 0.35
SLC6A2 P23975 2/20 0.35
HRH2 P25021 2/20 0.35
HTR2A P28223 2/20 0.35
SLC6A4 P31645 2/20 0.35
HRH1 P35367 2/20 0.35
SLC6A3 Q01959 2/20 0.35
KCNH2 Q12809 2/20 0.35
HRH3 Q9Y5N1 2/20 0.35
CYP2D6 P10635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4030524 0.87 MAOA (0.41) KMT2AP2RX7TSHR
SCHEMBL4032446 0.86 NFE2L2 (0.36) NFE2L2
SCHEMBL4038579 0.81 TRPA1 (0.39) TRPA1FFAR2MEN1KMT2AP2RX7
SCHEMBL2085063 0.78 GABRA1 (0.42) SLC6A2CYP2C9
SCHEMBL4038116 0.77 L3MBTL1 (0.40) TRPA1FFAR2MEN1KMT2AP2RX7
SCHEMBL4030343 0.73 TRPA1 (0.38) TRPA1FFAR2MEN1KMT2AP2RX7
SCHEMBL4031836 0.73 NPSR1 (0.34) NFE2L2CYP2C9LMNANPSR1
SCHEMBL6115316 0.72 TRIM24 (0.39) MEN1KMT2AL3MBTL1HTR1ALMNA
SCHEMBL31256727 0.72 TRPA1 (0.39) TRPA1FFAR2MEN1KMT2ANFE2L2
SCHEMBL3823757 0.71 TRIM24 (0.38) MEN1KMT2ANFE2L2TSHRL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed