SCHEMBL4038879

SCHEMBL4038879

CN(C)CCOCc1cc2c(s1)-c1cc(F)ccc1Sc1ccccc1-2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 5/20 0.38
DRD2 P14416 5/20 0.38
DRD1 P21728 5/20 0.38
HRH1 P35367 5/20 0.38
DRD3 P35462 5/20 0.38
ADRA2C P18825 4/20 0.38
HTR2A P28223 4/20 0.38
HTR2C P28335 4/20 0.38
MLNR O43193 2/20 0.38
NR1I2 O75469 2/20 0.38
CHRM2 P08172 2/20 0.38
HTR1A P08908 2/20 0.38
ADORA3 P0DMS8 2/20 0.38
CHRM1 P11229 2/20 0.38
PTGS1 P23219 2/20 0.38
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38
ADRA1A P35348 2/20 0.38
OPRM1 P35372 2/20 0.38
MC3R P41968 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4036021 0.99 ADRA2A (0.37) ADRA2ADRD2DRD1HRH1DRD3
SCHEMBL4039813 0.94 MEN1 (0.35) ADRA2ADRD2DRD1HRH1DRD3
Hydrochloric Acid SCHEMBL4037401 0.93 MEN1 (0.36) ADRA2ADRD2DRD1HRH1DRD3
SCHEMBL6336135 0.93 RAD52 (0.39) ADRA2ADRD2DRD1HRH1DRD3
Hydrochloric Acid SCHEMBL4039720 0.89 CHRM2 (0.39) ADRA2ADRD2DRD1HRH1DRD3
SCHEMBL6333796 0.88 MLNR (0.38) ADRA2ADRD2DRD1HRH1DRD3
SCHEMBL4037224 0.87 DRD2 (0.52) ADRA2ADRD2DRD1HRH1DRD3
SCHEMBL4037482 0.87 CHRM2 (0.38) ADRA2ADRD2DRD1HRH1DRD3
SCHEMBL6331962 0.86 KMT2A (0.38) ADRA2ADRD2DRD1HRH1DRD3
Hydrochloric Acid SCHEMBL4039786 0.86 LMNA (0.51) ADRA2ADRD2DRD1HRH1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1284977-B1 THIENODIBENZOAZULENE COMPOUNDS AS TUMOR NECROSIS FACTOR INHIBITORS GLAXOSMITHKLINE ZAGREB (HR) 2009-06-24 EP claimed
EP-2057146-A1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2009-05-13 EP claimed
WO-2008042639-A1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2008-04-10 WO claimed
EP-2057146-A1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2009-05-13 EP disclosed
WO-2008042639-A1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2008-04-10 WO disclosed