SCHEMBL4041872

SCHEMBL4041872

CC(C)CC(NC(=O)Oc1cc2sccc2s1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1cccnc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 5/20 0.38
HCRTR2 O43614 1/20 0.38
HSD17B10 Q99714 1/20 0.36
KCNQ1 P51787 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
LMNA P02545 2/20 0.33
CLK1 P49759 2/20 0.33
MEN1 O00255 1/20 0.33
POLB P06746 1/20 0.33
KMT2A Q03164 1/20 0.33
ELOVL6 Q9H5J4 1/20 0.33
SMYD3 Q9H7B4 1/20 0.32
MAPK1 P28482 1/20 0.32
HTT P42858 1/20 0.32
MMP1 P03956 1/20 0.32
MMP3 P08254 1/20 0.32
MMP9 P14780 1/20 0.32
CTSL P07711 2/20 0.32
CTSB P07858 2/20 0.32
CTSS P25774 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043056 0.93 HSD17B10 (0.36) HCRTR2HSD17B10KCNQ1SMN1; SMN2LMNA
SCHEMBL4051011 0.92 HCRTR2 (0.34) HCRTR2HSD17B10KCNQ1SMN1; SMN2LMNA
SCHEMBL4044312 0.90 CTSK (0.40) CTSKHCRTR2HSD17B10KCNQ1SMN1; SMN2
SCHEMBL4039560 0.90 HCRTR2 (0.33) CTSKHCRTR2HSD17B10KCNQ1SMN1; SMN2
SCHEMBL4045303 0.90 CTSK (0.37) CTSKSMYD3CTSLCTSBCTSS
SCHEMBL4047331 0.90 CTSK (0.40) CTSKMMP1MMP3MMP9CTSL
SCHEMBL4049190 0.89 CTSK (0.40) CTSKHCRTR2HSD17B10KCNQ1KMT2A
SCHEMBL4049345 0.88 CTSK (0.38) CTSKCTSLCTSBCTSS
SCHEMBL4045875 0.87 CTSK (0.41) CTSKCTSLCTSBCTSS
SCHEMBL4042884 0.85 CTSK (0.41) CTSKMMP1MMP3MMP9CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed