SCHEMBL4045303

SCHEMBL4045303

CC(C)CC(NC(=O)Oc1cc2sccc2s1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSK P43235 8/20 0.37
SMYD3 Q9H7B4 2/20 0.34
CTSL P07711 5/20 0.33
CTSS P25774 3/20 0.33
CTSB P07858 2/20 0.33
ALDH1A1 P00352 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
FKBP1A P62942 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4044199 0.93 SMYD3 (0.34) SMYD3ALDH1A1FKBP1A
SCHEMBL4044323 0.92 SMYD3 (0.33) SMYD3FKBP1A
SCHEMBL4042904 0.91 CTSK (0.39) CTSKSMYD3CTSLCTSSCTSB
SCHEMBL4045954 0.91 SMYD3 (0.33) CTSKSMYD3CTSSCTSBALDH1A1
SCHEMBL4041872 0.90 CTSK (0.38) CTSKSMYD3CTSLCTSSCTSB
SCHEMBL4043196 0.89 CTSK (0.39) CTSKSMYD3CTSLCTSSCTSB
SCHEMBL4047331 0.88 CTSK (0.40) CTSKCTSLCTSSCTSB
SCHEMBL4051023 0.88 CTSK (0.39) CTSKCTSLCTSSCTSBALDH1A1
SCHEMBL4042884 0.87 CTSK (0.41) CTSKCTSLCTSSCTSBALDH1A1
SCHEMBL4044003 0.85 CTSK (0.40) CTSKCTSLCTSSCTSBFKBP1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed