SCHEMBL4042306

SCHEMBL4042306

CCCC(NC(=O)Oc1ccc(-c2ccccn2)s1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1ccccn1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MMP8 P22894 4/20 0.37
MMP3 P08254 3/20 0.37
ALDH1A1 P00352 1/20 0.35
CTSK P43235 4/20 0.34
MMP13 P45452 1/20 0.33
PREP P48147 1/20 0.33
FAP Q12884 1/20 0.33
CTSS P25774 1/20 0.33
MMP1 P03956 1/20 0.32
MMP2 P08253 1/20 0.32
MMP7 P09237 1/20 0.32
ELANE P08246 1/20 0.32
KMT2A Q03164 1/20 0.31
CHRNA7 P36544 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4044090 0.95 CTSK (0.34) MMP8MMP3ALDH1A1CTSKMMP13
SCHEMBL4042987 0.93 CTSK (0.41) MMP8MMP3ALDH1A1CTSKMMP13
SCHEMBL4043813 0.90 CHRNB2 (0.36) MMP8MMP3ALDH1A1CTSKCTSS
SCHEMBL4045076 0.90 ALDH1A1 (0.38) ALDH1A1CTSKCTSS
SCHEMBL4038257 0.88 PREP (0.34) ALDH1A1CTSKPREPFAPELANE
SCHEMBL4045022 0.88 CTSK (0.35) CTSKPREPFAPCTSSELANE
SCHEMBL4047432 0.88 ALDH1A1 (0.35) MMP8MMP3ALDH1A1CTSKMMP13
SCHEMBL4045898 0.87 CTSK (0.41) ALDH1A1CTSKCTSSELANEKMT2A
SCHEMBL4043638 0.87 ALDH1A1 (0.35) MMP3ALDH1A1CTSKMMP13PREP
SCHEMBL4043139 0.86 ELANE (0.37) MMP8MMP3ALDH1A1CTSKMMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed