SCHEMBL4043813

SCHEMBL4043813

CCCC(NC(=O)Oc1ccc(-c2ccccn2)s1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.36
CHRNA7 P36544 1/20 0.36
CHRNA4 P43681 1/20 0.36
MMP8 P22894 2/20 0.33
MMP3 P08254 1/20 0.33
ALDH1A1 P00352 1/20 0.33
FKBP1A P62942 1/20 0.33
SMYD3 Q9H7B4 2/20 0.32
CTSK P43235 2/20 0.32
CTSS P25774 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043393 0.93 FKBP1A (0.35) CHRNB2CHRNA7CHRNA4FKBP1ASMYD3
SCHEMBL4043638 0.90 ALDH1A1 (0.35) CHRNB2CHRNA7CHRNA4MMP3ALDH1A1
SCHEMBL4042306 0.90 MMP8 (0.37) CHRNA7MMP8MMP3ALDH1A1CTSK
SCHEMBL4046884 0.89 CTSK (0.34) CHRNB2CHRNA7CHRNA4MMP3ALDH1A1
SCHEMBL4042787 0.88 CHRNB2 (0.37) CHRNB2CHRNA7CHRNA4ALDH1A1CTSK
SCHEMBL4045076 0.87 ALDH1A1 (0.38) ALDH1A1CTSKCTSS
SCHEMBL4040719 0.86 SMYD3 (0.35) ALDH1A1FKBP1ASMYD3CTSKCTSS
SCHEMBL4050153 0.86 SMYD3 (0.35) ALDH1A1FKBP1ASMYD3
SCHEMBL4044003 0.86 CTSK (0.40) CHRNB2CHRNA7CHRNA4FKBP1ACTSK
SCHEMBL4044090 0.85 CTSK (0.34) MMP8MMP3ALDH1A1CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed