SCHEMBL4047432

SCHEMBL4047432

CCCC(NC(=O)Oc1ccc(-c2ccccn2)s1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)C(=O)c1ccccn1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
CTSK P43235 3/20 0.34
MMP13 P45452 1/20 0.33
PREP P48147 1/20 0.33
FAP Q12884 1/20 0.33
MMP8 P22894 2/20 0.32
MMP3 P08254 2/20 0.32
MMP1 P03956 1/20 0.32
MMP2 P08253 1/20 0.32
MMP7 P09237 1/20 0.32
CTSS P25774 1/20 0.31
CHRNA7 P36544 2/20 0.31
NPY5R Q15761 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4039641 0.95 CTSK (0.34) CTSKPREPFAP
SCHEMBL4045577 0.93 CTSK (0.41) ALDH1A1CTSKMMP13MMP8MMP3
SCHEMBL4046884 0.91 CTSK (0.34) ALDH1A1CTSKMMP13PREPFAP
SCHEMBL4045076 0.90 ALDH1A1 (0.38) ALDH1A1CTSKCTSS
SCHEMBL6216815 0.89 CHRNA7 (0.39) ALDH1A1CTSKPREPFAPCTSS
SCHEMBL4045685 0.88 PREP (0.34) CTSKPREPFAP
SCHEMBL4042306 0.88 MMP8 (0.37) ALDH1A1CTSKMMP13PREPFAP
SCHEMBL4043203 0.88 CTSK (0.35) ALDH1A1CTSKPREPFAPCTSS
SCHEMBL4043638 0.87 ALDH1A1 (0.35) ALDH1A1CTSKMMP13PREPFAP
SCHEMBL4044691 0.86 PREP (0.35) CTSKPREPFAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed