SCHEMBL4043670

SCHEMBL4043670

O=C(NC(CC1CCCCC1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1cccnc1)Oc1csc2ccccc12

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSV O60911 2/20 0.37
CTSL P07711 2/20 0.37
CTSS P25774 2/20 0.37
F12 P00748 5/20 0.35
KCNQ1 P51787 1/20 0.35
ALDH1A1 P00352 1/20 0.34
GCK P35557 2/20 0.33
HSD17B10 Q99714 1/20 0.33
CALCRL Q16602 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4044172 0.91 CTSS (0.36) CTSVCTSLCTSSF12GCK
SCHEMBL4048072 0.91 CTSV (0.39) CTSVCTSLCTSSF12CALCRL
SCHEMBL4052140 0.90 HSD17B10 (0.36) KCNQ1ALDH1A1HSD17B10TSHR
SCHEMBL4214125 0.90 CTSS (0.38) CTSVCTSLCTSSF12GCK
SCHEMBL4039394 0.88 CTSL (0.42) CTSVCTSLCTSSF12GCK
SCHEMBL4049892 0.86 CTSS (0.37) CTSVCTSLCTSSF12GCK
SCHEMBL4045088 0.86 CTSS (0.37) CTSVCTSLCTSSF12CALCRL
SCHEMBL4046543 0.85 KCNQ1 (0.38) CTSVCTSLCTSSF12KCNQ1
SCHEMBL4048674 0.85 CTSS (0.37) CTSVCTSLCTSSF12GCK
SCHEMBL4043598 0.84 CTSS (0.37) CTSVCTSLCTSSF12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed