SCHEMBL4043596

SCHEMBL4043596

CCCC(NC(=O)Oc1ccc(-c2ccccc2)cc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)C(=O)c1cccnc1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ELANE P08246 1/20 0.38
CTSK P43235 5/20 0.37
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C9 P11712 2/20 0.35
TSHR P16473 1/20 0.35
ALDH1A1 P00352 1/20 0.34
GPR132 Q9UNW8 3/20 0.33
MMP1 P03956 1/20 0.32
MMP3 P08254 1/20 0.32
MMP9 P14780 1/20 0.32
PREP P48147 2/20 0.32
FAP Q12884 2/20 0.32
CYP2C19 P33261 1/20 0.32
CCR1 P32246 1/20 0.32
MC4R P32245 1/20 0.32
MC3R P41968 1/20 0.32
MC1R Q01726 1/20 0.32
TGM2 P21980 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4045571 0.92 CTSK (0.46) ELANECTSKMMP1MMP3MMP9
SCHEMBL4051965 0.92 MC4R (0.38) ELANECTSKCYP3A4CYP2C9ALDH1A1
SCHEMBL4048312 0.89 KCNQ1 (0.40) ELANECTSKTSHRALDH1A1
SCHEMBL4044808 0.89 CTSK (0.36) ELANECTSKCYP1A2CYP3A4CYP2C9
SCHEMBL4042585 0.89 USP30 (0.39) ELANECTSKTSHRALDH1A1MC4R
SCHEMBL4045553 0.89 CTSK (0.34) ELANECTSKALDH1A1GPR132PREP
SCHEMBL4051473 0.89 CTSK (0.34) ELANECTSKALDH1A1GPR132PREP
SCHEMBL4042529 0.89 BCL2 (0.38) ELANECTSKGPR132MC4RMC3R
SCHEMBL4042885 0.88 TGM2 (0.44) CTSKTGM2
SCHEMBL4044339 0.88 ALDH1A1 (0.37) ELANECTSKALDH1A1GPR132MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed