SCHEMBL4042585

SCHEMBL4042585

COc1ccc(CC(NC(=O)Oc2ccc(-c3ccccc3)cc2)C(=O)N2CCC3C2C(=O)CN3S(=O)(=O)C(=O)c2cccnc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 1/20 0.39
ITGA4 P13612 9/20 0.38
ITGB7 P26010 9/20 0.38
CTSK P43235 2/20 0.37
BCL2 P10415 1/20 0.36
F2 P00734 2/20 0.36
ELANE P08246 1/20 0.36
ITGB3 P05106 1/20 0.36
ITGAV P06756 1/20 0.36
MC4R P32245 1/20 0.36
MC3R P41968 1/20 0.36
MC1R Q01726 1/20 0.36
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
TSHR P16473 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4042529 0.94 BCL2 (0.38) ITGA4ITGB7CTSKBCL2ELANE
SCHEMBL4043465 0.93 MC4R (0.41) ITGA4ITGB7CTSKBCL2ELANE
SCHEMBL4045571 0.90 CTSK (0.46) CTSKELANE
SCHEMBL4045597 0.90 ACE (0.36) CTSKBCL2F2ELANEMC4R
SCHEMBL4043596 0.89 ELANE (0.38) CTSKELANEMC4RMC3RMC1R
SCHEMBL4045511 0.89 F2 (0.38) ITGA4ITGB7CTSKF2ITGB3
SCHEMBL4045924 0.88 USP30 (0.40) USP30ITGA4ITGB7ITGB3ITGAV
SCHEMBL4041797 0.86 CTSK (0.50) USP30CTSKF2MC4RMC3R
SCHEMBL6213140 0.85 CTSK (0.44) CTSKBCL2ITGB3MC4RMC3R
SCHEMBL4046868 0.84 ITGB1 (0.37) ITGA4ITGB7CTSKBCL2F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed