SCHEMBL4045577

SCHEMBL4045577

CC(C)CC(NC(=O)Oc1ccc(-c2ccccn2)s1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)C(=O)c1ccccn1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSK P43235 13/20 0.41
CTSL P07711 9/20 0.34
CTSS P25774 8/20 0.34
CTSB P07858 3/20 0.34
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 2/20 0.33
MMP13 P45452 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HSD17B10 Q99714 1/20 0.33
KMT2A Q03164 1/20 0.33
MMP8 P22894 2/20 0.33
MMP3 P08254 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4047432 0.93 ALDH1A1 (0.35) CTSKCTSSALDH1A1MMP13MMP8
SCHEMBL4042672 0.91 CTSK (0.41) CTSKCTSLCTSSCTSBALDH1A1
SCHEMBL4042338 0.90 CTSK (0.43) CTSKCTSLCTSSCTSBALDH1A1
SCHEMBL4045960 0.88 CTSK (0.41) CTSKCTSLCTSSCTSBALDH1A1
SCHEMBL4045748 0.88 CTSK (0.51) CTSKCTSLCTSSCTSBALDH1A1
SCHEMBL4048011 0.88 CTSK (0.40) CTSKCTSLCTSSCTSB
SCHEMBL4042987 0.88 CTSK (0.41) CTSKCTSLCTSSCTSBALDH1A1
SCHEMBL4039641 0.87 CTSK (0.34) CTSK
SCHEMBL4046924 0.86 CTSK (0.40) CTSKCTSLCTSSCTSBALDH1A1
SCHEMBL4050151 0.86 CTSK (0.41) CTSKCTSLCTSSCTSBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed