SCHEMBL4046060

SCHEMBL4046060

CCCC(NC(=O)Oc1cccs1)C(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 4/20 0.35
PAX8 Q06710 1/20 0.34
ACACB O00763 1/20 0.33
GPR132 Q9UNW8 3/20 0.32
MAPT P10636 2/20 0.32
TSHR P16473 1/20 0.32
TNKS O95271 1/20 0.32
PARP1 P09874 1/20 0.32
PARP2 Q9UGN5 1/20 0.32
PARP4 Q9UKK3 1/20 0.32
PARP3 Q9Y6F1 1/20 0.32
CHRNA7 P36544 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
PREP P48147 1/20 0.32
FAP Q12884 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPK8 P45983 1/20 0.32
VNN1 O95497 1/20 0.32
F2 P00734 1/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4038998 0.92 CTSK (0.44) CTSKPAX8CHRNA7ALDH1A1
SCHEMBL4038641 0.89 CTSK (0.33) CTSKPAX8ACACBGPR132TNKS
SCHEMBL4045728 0.89 CTSK (0.35) CTSKPAX8ACACBGPR132TNKS
SCHEMBL4043616 0.87 CTSK (0.35) CTSKPAX8GPR132L3MBTL1PREP
SCHEMBL4044586 0.87 CTSK (0.37) CTSKPAX8GPR132TNKSPARP1
SCHEMBL4047771 0.87 CTSK (0.39) CTSKACACBGPR132CHRNA7
SCHEMBL4050153 0.86 SMYD3 (0.35) MAPTTSHRF2ALDH1A1
SCHEMBL4041663 0.86 CTSK (0.35) CTSKPAX8ACACBGPR132TSHR
SCHEMBL4047976 0.86 CTSK (0.43) CTSK
SCHEMBL4040981 0.86 CTSK (0.35) CTSKPAX8ACACBGPR132TNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed