SCHEMBL4043616

SCHEMBL4043616

CCCC(NC(=O)Oc1cc2ccccc2s1)C(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSK P43235 7/20 0.35
PAX8 Q06710 1/20 0.34
CYP3A4 P08684 1/20 0.33
PREP P48147 1/20 0.33
FAP Q12884 1/20 0.33
HTRA1 Q92743 1/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
ALDH1A1 P00352 1/20 0.33
GPR132 Q9UNW8 3/20 0.32
MMP1 P03956 1/20 0.32
MMP3 P08254 1/20 0.32
MMP9 P14780 1/20 0.32
DRD2 P14416 1/20 0.32
DRD3 P35462 1/20 0.32
BCHE P06276 1/20 0.32
ACHE P22303 1/20 0.32
TACR1 P25103 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050975 0.92 CTSK (0.43) CTSKPAX8ALDH1A1MMP1MMP3
SCHEMBL4038641 0.91 CTSK (0.33) CTSKPAX8PREPFAPL3MBTL1
SCHEMBL4043031 0.89 HTRA1 (0.37) CTSKPAX8HTRA1GPR132MMP1
SCHEMBL4044586 0.88 CTSK (0.37) CTSKPAX8PREPFAPGPR132
SCHEMBL4046060 0.87 CTSK (0.35) CTSKPAX8PREPFAPL3MBTL1
SCHEMBL4040719 0.87 SMYD3 (0.35) CTSKPREPFAPL3MBTL1ALDH1A1
SCHEMBL4046786 0.86 CHRNB2 (0.36) CTSKPAX8PREPFAPHTRA1
SCHEMBL4041238 0.86 CHRNB2 (0.36) CTSKPAX8PREPFAPHTRA1
SCHEMBL4047771 0.86 CTSK (0.39) CTSKGPR132
SCHEMBL4042787 0.86 CHRNB2 (0.37) CTSKPAX8PREPFAPALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed