SCHEMBL4044586

SCHEMBL4044586

CCCC(NC(=O)Oc1ccc(-c2ccccc2)s1)C(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSK P43235 7/20 0.37
CHRNB2 P17787 1/20 0.36
CHRNA7 P36544 1/20 0.36
CHRNA4 P43681 1/20 0.36
GPR132 Q9UNW8 3/20 0.34
CTSS P25774 1/20 0.33
PAX8 Q06710 2/20 0.33
SIGMAR1 Q99720 1/20 0.33
P2RX7 Q99572 1/20 0.32
TNKS O95271 1/20 0.32
PARP1 P09874 1/20 0.32
PARP2 Q9UGN5 1/20 0.32
PARP4 Q9UKK3 1/20 0.32
PARP3 Q9Y6F1 1/20 0.32
PREP P48147 1/20 0.32
FAP Q12884 1/20 0.32
MMP1 P03956 1/20 0.32
ACE P12821 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4042787 0.93 CHRNB2 (0.37) CTSKCHRNB2CHRNA7CHRNA4GPR132
SCHEMBL4045035 0.92 CTSK (0.45) CTSKCHRNB2CHRNA7CHRNA4CTSS
SCHEMBL4047771 0.89 CTSK (0.39) CTSKCHRNA7GPR132SIGMAR1
SCHEMBL4043616 0.88 CTSK (0.35) CTSKGPR132PAX8PREPFAP
SCHEMBL4046060 0.87 CTSK (0.35) CTSKCHRNA7GPR132PAX8TNKS
SCHEMBL4043393 0.87 FKBP1A (0.35) CTSKCHRNB2CHRNA7CHRNA4CTSS
SCHEMBL4047976 0.86 CTSK (0.43) CTSKCTSS
SCHEMBL4048981 0.85 CTSK (0.43) CTSKCHRNB2CHRNA7CHRNA4CTSS
SCHEMBL4038641 0.85 CTSK (0.33) CTSKGPR132PAX8TNKSPARP1
SCHEMBL4039018 0.85 HSD17B10 (0.36) CTSKCHRNB2CHRNA7CHRNA4CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed