SCHEMBL4046098

SCHEMBL4046098

CC(C)CC(NC(=O)Oc1ccc2c(c1)OCO2)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1cccc[n+]1[O-]

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSK P43235 10/20 0.39
LMNA P02545 2/20 0.36
PKM P14618 1/20 0.36
TSHR P16473 2/20 0.34
ALDH1A1 P00352 2/20 0.34
HPGD P15428 1/20 0.34
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
CTSL P07711 4/20 0.33
CTSS P25774 3/20 0.33
CTSB P07858 2/20 0.33
KCNQ1 P51787 1/20 0.32
KDM4E B2RXH2 1/20 0.32
POLB P06746 1/20 0.32
MCHR1 Q99705 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050306 0.93 PKM (0.36) CTSKLMNAPKMTSHRALDH1A1
SCHEMBL4047459 0.89 CTSK (0.38) CTSKLMNATSHRALDH1A1HPGD
SCHEMBL4047763 0.88 CTSK (0.44) CTSKCTSLCTSSCTSB
SCHEMBL4052113 0.86 CTSK (0.41) CTSKCTSLCTSSCTSB
SCHEMBL4045230 0.85 CTSK (0.43) CTSKCTSLCTSSCTSB
SCHEMBL4047523 0.85 CTSK (0.39) CTSKALDH1A1TAS1R3TAS1R1CTSL
SCHEMBL4044439 0.84 CTSK (0.41) CTSKCTSLCTSSCTSB
SCHEMBL4049409 0.83 CTSK (0.42) CTSKCTSLCTSSCTSB
SCHEMBL4046660 0.83 HTT (0.40) CTSKLMNATSHRALDH1A1HPGD
SCHEMBL4041781 0.83 CTSK (0.39) CTSKTAS1R3TAS1R1CTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed