SCHEMBL4050306

SCHEMBL4050306

CCCC(NC(=O)Oc1ccc2c(c1)OCO2)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1cccc[n+]1[O-]

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.36
TSHR P16473 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 1/20 0.35
LMNA P02545 2/20 0.34
CHRM5 P08912 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
EDNRB P24530 1/20 0.32
EDNRA P25101 1/20 0.32
KCNQ1 P51787 1/20 0.32
F2 P00734 3/20 0.32
F10 P00742 2/20 0.32
BMP1 P13497 1/20 0.32
ELANE P08246 1/20 0.32
KDM4E B2RXH2 1/20 0.32
POLB P06746 1/20 0.32
CTSK P43235 2/20 0.32
MCHR1 Q99705 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4046098 0.93 CTSK (0.39) PKMTSHRALDH1A1HPGDLMNA
SCHEMBL4049558 0.90 CTSK (0.36) F2F10ELANECTSK
SCHEMBL4048294 0.89 ALDH1A1 (0.37) TSHRALDH1A1HPGDLMNACHRM5
SCHEMBL4041133 0.88 CTSK (0.36) ALDH1A1F2F10ELANECTSK
SCHEMBL4044073 0.86 CTSK (0.33) F2F10CTSK
SCHEMBL4051941 0.85 ELOVL6 (0.38) TSHRLMNACTSK
SCHEMBL4048186 0.85 ALDH1A1 (0.36) ALDH1A1LMNACHRM5KDM4ECTSK
SCHEMBL4045941 0.85 CTSK (0.33) F2F10CTSK
SCHEMBL4046418 0.84 CTSK (0.33) F2F10CTSK
SCHEMBL4044424 0.84 CTSK (0.34) F2F10CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed