SCHEMBL4046172

SCHEMBL4046172

c1cnc2[nH]c(CCC3CC3)nc2n1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 1/20 0.35
METAP1 P53582 1/20 0.35
DRD2 P14416 1/20 0.34
DRD4 P21917 1/20 0.34
DRD3 P35462 1/20 0.34
CCNB2 O95067 1/20 0.31
CDK1 P06493 1/20 0.31
CCNB1 P14635 1/20 0.31
GSK3A P49840 1/20 0.31
GSK3B P49841 1/20 0.31
CCNB3 Q8WWL7 1/20 0.31
PBK Q96KB5 1/20 0.31
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4046851 0.94 LMNA (0.34) METAP2METAP1DRD2DRD4DRD3
SCHEMBL4047661 0.83 PBK (0.42) METAP2METAP1CCNB2CDK1CCNB1
SCHEMBL4040136 0.77 AAK1 (0.43) METAP2METAP1CCNB2CDK1CCNB1
SCHEMBL4052252 0.75 KDM4C (0.41) METAP2METAP1CCNB2CDK1CCNB1
SCHEMBL4047123 0.75 METAP2 (0.36) METAP2METAP1
SCHEMBL4051241 0.72 PI4KA (0.45) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL4044144 0.72 METAP2 (0.34) METAP2METAP1
SCHEMBL4046923 0.71 PI4KA (0.51) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL4046994 0.71 ADORA1 (0.42) METAP2METAP1CDK1CCNB1GSK3A
SCHEMBL4053122 0.69 GPR84 (0.47) METAP2METAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009029592-A1 HETEROBICYCLIC-SUBSTITUTED QUINOLONES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2009-03-05 WO disclosed
WO-2009029592-A1 HETEROBICYCLIC-SUBSTITUTED QUINOLONES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2009-03-05 WO disclosed