SCHEMBL4046460

SCHEMBL4046460

CON(C)C(=O)c1ccc(C2CCCCN2C(=O)C(F)(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 1/20 0.44
RIPK1 Q13546 4/20 0.43
ROCK2 O75116 5/20 0.38
SCD5 Q86SK9 1/20 0.38
HSD17B10 Q99714 1/20 0.37
CCNC P24863 1/20 0.37
CDK8 P49336 1/20 0.37
GPR119 Q8TDV5 2/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
PARP14 Q460N5 1/20 0.36
PARP10 Q53GL7 1/20 0.36
CFB P00751 1/20 0.35
EPHX2 P34913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4046089 0.82 RIPK1 (0.50) RIPK1ROCK2CCNCCDK8GAA
SCHEMBL4046232 0.80 RIPK1 (0.51) RIPK1CCNCCDK8GAAHPGD
SCHEMBL4051349 0.76 RIPK1 (0.44) RIPK1CCNCCDK8GAAHPGD
SCHEMBL28171621 0.76 RIPK1 (0.67) RIPK1SCD5PARP14PARP10EPHX2
SCHEMBL30878611 0.73 RIPK1 (0.55) RIPK1SCD5HSD17B10
SCHEMBL27564986 0.73 RIPK1 (0.62) RIPK1SCD5EPHX2
SCHEMBL1576663 0.72 RIPK1 (0.73) RIPK1SCD5EPHX2
SCHEMBL28916713 0.70 RIPK1 (0.48) RIPK1ROCK2HSD17B10GAAHPGD
SCHEMBL2576253 0.70 MLYCD (0.50) MLYCDGPR119HPGD
SCHEMBL5458875 0.69 NPC1 (0.48) RIPK1HSD17B10GAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009103478-A1 PYRIDONE AND PYRIDAZINONE DERIVATIVES AS MCH ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-08-27 WO disclosed