SCHEMBL4048343

SCHEMBL4048343

COc1cc(OC)cc(N2C(N)=NN(c3nccs3)C2N)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP1A1 P04798 4/20 0.33
CYP1A2 P05177 4/20 0.33
CYP1B1 Q16678 4/20 0.33
TP53 P04637 2/20 0.33
SRC P12931 1/20 0.33
ZAP70 P43403 1/20 0.33
SYK P43405 1/20 0.33
MDM2 Q00987 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
HPGD P15428 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
ATM Q13315 1/20 0.32
HSD17B10 Q99714 1/20 0.32
UBE2I P63279 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4038866 0.89 SRC (0.39) NPC1RAB9AMEN1KMT2ASRC
SCHEMBL4036701 0.85 HTT (0.36) MEN1KMT2ASMN1; SMN2HPGDKDM4E
SCHEMBL4043372 0.60 ZAP70 (0.50) CYP1A1CYP1A2CYP1B1SRCZAP70
SCHEMBL4048336 0.60 CYP1A1 (0.46) NPC1RAB9ACYP1A1CYP1A2CYP1B1
SCHEMBL31374372 0.60 NPC1 (0.47) NPC1RAB9AMEN1KMT2ACYP1A2
SCHEMBL28257980 0.57 ROCK1 (0.55) NPC1RAB9AMEN1KMT2AHPGDS
Anisole SCHEMBL28150475 0.57 ALDH1A1 (0.56) NPC1RAB9AMEN1KMT2ACYP1A1
SCHEMBL6319123 0.56 GABRA1 (0.45) NPC1RAB9AMEN1KMT2ACYP1A1
SCHEMBL4895926 0.55 GABRA1 (0.44) NPC1RAB9AMEN1KMT2ACYP1A1
SCHEMBL14675928 0.54 KMT2A (0.56) NPC1RAB9AMEN1KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562589-B1 DIAMINOTRIAZOLES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2009-01-07 EP disclosed