SCHEMBL4038866

SCHEMBL4038866

COc1cc(N2C(N)=NN(c3nccs3)C2N)cc(C(F)(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 3/20 0.39
ZAP70 P43403 3/20 0.39
SYK P43405 3/20 0.39
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
KDM1A O60341 1/20 0.35
DPP4 P27487 2/20 0.35
CTSD P07339 3/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
FGFR2 P21802 1/20 0.32
FGFR3 P22607 1/20 0.32
PHGDH O43175 1/20 0.32
CDK4 P11802 1/20 0.30
CDK2 P24941 1/20 0.30
PDE10A Q9Y233 1/20 0.30
HDAC3 O15379 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4048343 0.89 NPC1 (0.42) SRCZAP70SYKNPC1RAB9A
SCHEMBL4036701 0.78 HTT (0.36) MEN1KMT2A
SCHEMBL4038860 0.65 SRC (0.52) SRCZAP70SYKCDK4CDK2
SCHEMBL4039114 0.65 SRC (0.56) SRCZAP70SYKCDK4CDK2
SCHEMBL788369 0.60 DPP4 (0.39) KDM1ADPP4MEN1KMT2APHGDH
SCHEMBL679095 0.59 ALDH1A1 (0.50) RAB9AKDM1ADPP4HDAC3HDAC1
SCHEMBL5782136 0.59 ALDH1A1 (0.58) RAB9AKDM1AHDAC3HDAC1HDAC2
SCHEMBL8333311 0.59 CYP11B1 (0.55) MEN1KMT2A
SCHEMBL130736 0.58 L3MBTL1 (0.45) RAB9AKDM1ADPP4HDAC3HDAC1
SCHEMBL30448494 0.58 L3MBTL1 (0.45) RAB9AKDM1ADPP4HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562589-B1 DIAMINOTRIAZOLES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2009-01-07 EP disclosed