SCHEMBL4036701

SCHEMBL4036701

Cc1cc(C)cc(N2C(N)=NN(c3nccs3)C2N)c1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.36
TDP1 Q9NUW8 2/20 0.33
ALDH1A1 P00352 4/20 0.31
MAPT P10636 3/20 0.31
KDM4E B2RXH2 2/20 0.31
GFER P55789 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
POLB P06746 1/20 0.31
APEX1 P27695 1/20 0.31
RECQL P46063 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
NPSR1 Q6W5P4 2/20 0.30
GAA P10253 1/20 0.30
MEN1 O00255 1/20 0.30
HPGD P15428 1/20 0.30
KMT2A Q03164 1/20 0.30
TSHR P16473 1/20 0.30
NOS1 P29475 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4048343 0.85 NPC1 (0.42) TDP1ALDH1A1KDM4ESMN1; SMN2POLB
SCHEMBL4042829 0.78 NOS1 (0.34) NOS1
SCHEMBL4038866 0.78 SRC (0.39) MEN1KMT2A
SCHEMBL27398935 0.56 SMPD3 (0.46) ALDH1A1RECQLTSHRNOS1HSD17B10
SCHEMBL28145280 0.56 ALDH1A1 (0.39) TDP1ALDH1A1KDM4EPOLBAPEX1
Bromide SCHEMBL28899538 0.56 TDP1 (0.37) TDP1ALDH1A1MAPTKDM4EPOLB
SCHEMBL2857147 0.56 NPC1 (0.41) HTTTDP1ALDH1A1POLBAPEX1
SCHEMBL16549064 0.56 LMNA (0.43) MAPTKDM4EGFERSMN1; SMN2POLB
SCHEMBL28830908 0.55 TDP1 (0.54) TDP1ALDH1A1MAPTKDM4ESMN1; SMN2
SCHEMBL29261700 0.55 KDM4E (0.42) TDP1ALDH1A1MAPTKDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562589-B1 DIAMINOTRIAZOLES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2009-01-07 EP disclosed