SCHEMBL4048550

SCHEMBL4048550

CCCCC(CC)c1nc2nccnc2[nH]1

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 3/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33
METAP2 P50579 1/20 0.33
METAP1 P53582 1/20 0.33
KDM4E B2RXH2 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ALDH1A1 P00352 2/20 0.30
CYP3A4 P08684 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4054698 0.87 ADORA3 (0.40) ADORA3ADORA2AADORA2BADORA1METAP2
SCHEMBL4047234 0.83 GPR84 (0.43) METAP2METAP1ALDH1A1
SCHEMBL11830439 0.82 TSHR (0.34) ADORA3ADORA2AADORA2BADORA1ALDH1A1
SCHEMBL22962317 0.74 PDE5A (0.48) METAP2METAP1SMN1; SMN2ALDH1A1
SCHEMBL22961994 0.73 TLR8 (0.39) ADORA3KDM4ESMN1; SMN2ALDH1A1
SCHEMBL22962333 0.73 AURKA (0.39) ADORA3ADORA2AADORA2BADORA1
SCHEMBL4043723 0.71 METAP2 (0.41) ADORA3ADORA2AADORA2BADORA1METAP2
SCHEMBL22962315 0.70 ADORA3 (0.34) ADORA3ADORA2AADORA2BADORA1KDM4E
SCHEMBL5088882 0.69 CYP1A2 (0.41) SMN1; SMN2ALDH1A1CYP3A4
SCHEMBL18923160 0.69 CYP1A2 (0.41) SMN1; SMN2ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009029592-A1 HETEROBICYCLIC-SUBSTITUTED QUINOLONES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2009-03-05 WO disclosed