SCHEMBL4054698

SCHEMBL4054698

CCC(CC)c1nc2nccnc2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
ADORA1 P30542 1/20 0.40
METAP2 P50579 1/20 0.38
METAP1 P53582 1/20 0.38
EGLN1 Q9GZT9 1/20 0.31
KDM4E B2RXH2 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4048550 0.87 ADORA3 (0.33) ADORA3ADORA2AADORA2BADORA1METAP2
SCHEMBL4048043 0.84 METAP2 (0.37) METAP2METAP1EGLN1
SCHEMBL4043723 0.79 METAP2 (0.41) ADORA3ADORA2AADORA2BADORA1METAP2
SCHEMBL4046285 0.77 GPR84 (0.35) METAP2METAP1KDM4ESMN1; SMN2
SCHEMBL4048086 0.76 METAP2 (0.39) METAP2METAP1EGLN1
SCHEMBL4047234 0.75 GPR84 (0.43) METAP2METAP1
SCHEMBL3951248 0.74 ADORA3 (0.38) ADORA3ADORA2AADORA2BADORA1KDM4E
SCHEMBL3948888 0.73 ADORA3 (0.34) ADORA3ADORA2AADORA2BADORA1KDM4E
SCHEMBL4052403 0.71 METAP2 (0.36) METAP2METAP1EGLN1
SCHEMBL13905132 0.71 METAP2 (0.33) METAP2METAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009029592-A1 HETEROBICYCLIC-SUBSTITUTED QUINOLONES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2009-03-05 WO disclosed