SCHEMBL4049689

SCHEMBL4049689

Cc1ccc(CC2(N(C)C)CCC(NC(=O)CCCC(=O)c3ccccc3)CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.53
MEN1 O00255 3/20 0.53
CCR2 P41597 3/20 0.48
OPRM1 P35372 2/20 0.43
OPRL1 P41146 2/20 0.43
KCNH2 Q12809 1/20 0.41
EPHX2 P34913 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
EPHX1 P07099 1/20 0.41
ADRA1D P25100 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
MCHR1 Q99705 1/20 0.40
HDAC1 Q13547 2/20 0.39
HDAC3 O15379 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4048631 0.94 KMT2A (0.51) KMT2AMEN1CCR2OPRM1OPRL1
SCHEMBL4054992 0.91 CCR2 (0.59) KMT2AMEN1CCR2OPRM1OPRL1
SCHEMBL206079 0.87 OPRM1 (0.54) OPRM1OPRL1EPHX2EPHX1
SCHEMBL4072325 0.85 OPRM1 (0.52) OPRM1OPRL1EPHX2EPHX1
SCHEMBL4048579 0.84 KMT2A (0.47) KMT2AMEN1CCR2OPRM1OPRL1
SCHEMBL4048586 0.84 CCR2 (0.49) KMT2AMEN1CCR2OPRM1OPRL1
SCHEMBL2976452 0.84 MEN1 (0.46) KMT2AMEN1OPRM1OPRL1RAB9A
SCHEMBL4054571 0.84 ACKR3 (0.49) KMT2AMEN1MCHR1
SCHEMBL4049886 0.84 MAPT (0.45) KMT2AMEN1CCR2NPC1RAB9A
SCHEMBL4052851 0.83 KMT2A (0.48) KMT2AMEN1OPRM1OPRL1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7476763-B2 Oxo-substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2009-01-13 US disclosed