SCHEMBL4048586

SCHEMBL4048586

CN(C)C1(Cc2cccc(Cl)c2)CCC(NC(=O)CCCC(=O)c2ccccc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 4/20 0.49
THRB P10828 1/20 0.47
HPGD P15428 1/20 0.47
SIGMAR1 Q99720 1/20 0.45
EPHX2 P34913 2/20 0.45
KCNH2 Q12809 1/20 0.43
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
POLB P06746 1/20 0.42
OPRM1 P35372 1/20 0.42
OPRL1 P41146 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
EPHX1 P07099 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4054992 0.89 CCR2 (0.59) CCR2HPGDSIGMAR1EPHX2KCNH2
SCHEMBL2977995 0.87 THRB (0.48) THRBHPGDSIGMAR1EPHX2KMT2A
SCHEMBL4048483 0.86 SIGMAR1 (0.48) THRBHPGDSIGMAR1EPHX2KMT2A
SCHEMBL16143720 0.85 SIGMAR1 (0.44) THRBHPGDSIGMAR1EPHX2OPRM1
SCHEMBL4049689 0.84 KMT2A (0.53) CCR2EPHX2KCNH2KMT2AMEN1
SCHEMBL206966 0.84 EPHX2 (0.62) THRBHPGDSIGMAR1EPHX2KMT2A
SCHEMBL206079 0.84 OPRM1 (0.54) SIGMAR1EPHX2OPRM1OPRL1EPHX1
SCHEMBL4052851 0.83 KMT2A (0.48) KMT2AMEN1OPRM1OPRL1
SCHEMBL206084 0.83 EPHX2 (0.47) THRBHPGDSIGMAR1EPHX2OPRM1
SCHEMBL207910 0.83 OPRM1 (0.50) THRBHPGDSIGMAR1EPHX2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7476763-B2 Oxo-substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2009-01-13 US disclosed