SCHEMBL2976452

SCHEMBL2976452

COC(=O)CCCC(=O)NC1CCC(Cc2ccc(C)cc2)(N(C)C)CC1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
HPGD P15428 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
SMYD3 Q9H7B4 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRL1 P41146 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2989386 0.90 LMNA (0.45) HPGDCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL2982804 0.90 CYP1A2 (0.42) HPGDCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL2985381 0.90 OPRM1 (0.48) HPGDCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL2987319 0.88 MEN1 (0.47) MEN1KMT2AKDM4EOPRM1OPRL1
SCHEMBL2983415 0.87 MEN1 (0.45) MEN1KMT2AHPGDCYP1A2CYP3A4
SCHEMBL4049689 0.84 KMT2A (0.53) MEN1KMT2ARAB9AOPRM1OPRL1
SCHEMBL206079 0.83 OPRM1 (0.54) OPRM1OPRL1
SCHEMBL2983741 0.83 SIGMAR1 (0.41) MEN1KMT2AALDH1A1SMN1; SMN2OPRM1
SCHEMBL2977995 0.83 THRB (0.48) MEN1KMT2AHPGDSMN1; SMN2L3MBTL1
SCHEMBL5162372 0.82 RAB9A (0.43) MEN1KMT2AHPGDKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7786328-B2 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2010-08-31 US claimed
US-20070281954-A1 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2007-12-06 US claimed
US-7786328-B2 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2010-08-31 US disclosed
US-20070281954-A1 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2007-12-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070281954-A1 Cyclohexyl-1,4-diamine compounds DPYD, PKD1, AOC1 MEN1 318/4885KMT2A 3786/4885HPGD 162/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.