SCHEMBL4050866

SCHEMBL4050866

CC(C)CC(NC(=O)Oc1ccc2ccccc2n1)C(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSK P43235 13/20 0.43
CHRNB2 P17787 2/20 0.38
CHRNA7 P36544 2/20 0.38
CHRNA4 P43681 2/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CTSL P07711 7/20 0.37
CTSS P25774 5/20 0.37
CTSB P07858 4/20 0.37
ALDH1A1 P00352 1/20 0.36
MMP1 P03956 2/20 0.35
MMP3 P08254 2/20 0.35
MMP9 P14780 2/20 0.35
HTRA1 Q92743 1/20 0.34
PAX8 Q06710 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4041238 0.92 CHRNB2 (0.36) CTSKCHRNB2CHRNA7CHRNA4CHRNB4
SCHEMBL4048898 0.92 CTSK (0.43) CTSKCTSLCTSSCTSBALDH1A1
SCHEMBL4045179 0.89 CTSK (0.44) CTSKCHRNA7CTSLCTSSCTSB
SCHEMBL4051166 0.87 CTSK (0.39) CTSKCHRNB2CHRNA7CHRNA4CHRNB4
SCHEMBL4050975 0.86 CTSK (0.43) CTSKCTSLCTSSCTSBALDH1A1
SCHEMBL4045083 0.86 CTSK (0.47) CTSKCHRNA7CTSLCTSSCTSB
SCHEMBL4048629 0.85 CTSK (0.42) CTSKCTSLCTSSCTSBALDH1A1
SCHEMBL4042383 0.85 CTSK (0.42) CTSKCHRNB2CHRNA7CHRNA4CTSL
SCHEMBL4048929 0.85 CTSK (0.52) CTSKCTSLCTSSCTSB
SCHEMBL4039165 0.85 CTSK (0.40) CTSKCHRNB2CHRNA7CHRNA4CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed