SCHEMBL4050975

SCHEMBL4050975

CC(C)CC(NC(=O)Oc1cc2ccccc2s1)C(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSK P43235 14/20 0.43
CTSL P07711 6/20 0.37
CTSS P25774 4/20 0.37
CTSB P07858 2/20 0.37
MMP1 P03956 1/20 0.36
MMP3 P08254 1/20 0.36
MMP9 P14780 1/20 0.36
TAS1R3 Q7RTX0 2/20 0.36
TAS1R1 Q7RTX1 2/20 0.36
PAX8 Q06710 1/20 0.36
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043616 0.92 CTSK (0.35) CTSKMMP1MMP3MMP9PAX8
SCHEMBL4042884 0.90 CTSK (0.41) CTSKCTSLCTSSCTSBMMP1
SCHEMBL4045179 0.89 CTSK (0.44) CTSKCTSLCTSSCTSBMMP1
SCHEMBL4045035 0.88 CTSK (0.45) CTSKCTSLCTSSCTSBPAX8
SCHEMBL4038998 0.87 CTSK (0.44) CTSKCTSLCTSSCTSBPAX8
SCHEMBL4042904 0.87 CTSK (0.39) CTSKCTSLCTSSCTSBMMP1
SCHEMBL4042383 0.86 CTSK (0.42) CTSKCTSLCTSSCTSBMMP1
SCHEMBL4050866 0.86 CTSK (0.43) CTSKCTSLCTSSCTSBMMP1
SCHEMBL4045083 0.86 CTSK (0.47) CTSKCTSLCTSSCTSBMMP1
SCHEMBL4048981 0.86 CTSK (0.43) CTSKCTSLCTSSCTSBPAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed