SCHEMBL4041238

SCHEMBL4041238

CCCC(NC(=O)Oc1ccc2ccccc2n1)C(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.36
CHRNA7 P36544 2/20 0.36
CHRNA4 P43681 2/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CTSK P43235 6/20 0.35
PREP P48147 2/20 0.35
FAP Q12884 2/20 0.35
HTRA1 Q92743 1/20 0.34
PAX8 Q06710 1/20 0.33
P2RX7 Q99572 1/20 0.32
MC4R P32245 1/20 0.32
MC3R P41968 1/20 0.32
MC1R Q01726 1/20 0.32
MMP1 P03956 1/20 0.32
VNN1 O95497 1/20 0.32
ACACB O00763 1/20 0.31
HCRTR2 O43614 1/20 0.31
XIAP P98170 1/20 0.31
SIGMAR1 Q99720 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050866 0.92 CTSK (0.43) CHRNB2CHRNA7CHRNA4CHRNB4CHRNA3
SCHEMBL4045929 0.92 PREP (0.36) CTSKPREPFAPHTRA1PAX8
SCHEMBL4043031 0.89 HTRA1 (0.37) CHRNA7CTSKHTRA1PAX8MC4R
SCHEMBL4046652 0.87 CHRNB2 (0.35) CHRNB2CHRNA7CHRNA4CHRNB4CHRNA3
SCHEMBL4043616 0.86 CTSK (0.35) CTSKPREPFAPHTRA1PAX8
SCHEMBL4047771 0.86 CTSK (0.39) CHRNA7CTSKACACBSIGMAR1
SCHEMBL4044443 0.85 ALDH1A1 (0.38) CTSKPREPFAPHTRA1PAX8
SCHEMBL4046786 0.85 CHRNB2 (0.36) CHRNB2CHRNA7CHRNA4CTSKPREP
SCHEMBL4047976 0.85 CTSK (0.43) CTSK
SCHEMBL4048207 0.85 HSD17B10 (0.36) CHRNB2CHRNA7CHRNA4CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed