SCHEMBL4059484

SCHEMBL4059484

COC(=O)C1CC(C#N)(c2ccc(OC)c3c2c2cc(F)ccc2n3C)CCC1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 1/20 0.41
PSEN2 P49810 1/20 0.41
APH1B Q8WW43 1/20 0.41
NCSTN Q92542 1/20 0.41
APH1A Q96BI3 1/20 0.41
PSENEN Q9NZ42 1/20 0.41
ADRA2A P08913 3/20 0.33
ADRA2B P18089 3/20 0.33
ADRA2C P18825 3/20 0.33
ADRA1A P35348 3/20 0.33
HRH1 P35367 3/20 0.33
ADRA1D P25100 2/20 0.33
ADRA1B P35368 2/20 0.33
BACE1 P56817 1/20 0.33
BACE2 Q9Y5Z0 1/20 0.33
PDE4A P27815 4/20 0.33
PDE4B Q07343 4/20 0.33
PDE4C Q08493 4/20 0.33
PDE4D Q08499 4/20 0.33
KDM4E B2RXH2 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4051064 0.88 ALDH1A1 (0.34) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL13693820 0.84 PDE4A (0.41) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL4241620 0.79 PSEN1 (0.35) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4063486 0.79 MYLK (0.33) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL4058008 0.78 PDE4A (0.33) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL4054310 0.76 PDE10A (0.36) KDM4EPIN1HTR2AHTR2CHTR2B
SCHEMBL6617848 0.75 PDE4A (0.39) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL13693578 0.75 PIN1 (0.31) KDM4EPIN1
SCHEMBL1558214 0.74 RORC (0.45) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4012666 0.74 PDE4B (0.37) PDE4APDE4BPDE4CPDE4DKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO disclosed