SCHEMBL4051346

SCHEMBL4051346

CC(C)(C)CC(NC(=O)Oc1csc2ccccc12)C(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.38
PTGER2 P43116 5/20 0.33
PAX8 Q06710 1/20 0.32
CALCRL Q16602 1/20 0.31
F2 P00734 1/20 0.31
CTSB P07858 1/20 0.31
CTSS P25774 1/20 0.31
PTGER4 P35408 1/20 0.31
PTGER3 P43115 1/20 0.31
ALDH1A1 P00352 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
SIGMAR1 Q99720 1/20 0.30
TNKS O95271 1/20 0.30
PARP1 P09874 1/20 0.30
PARP2 Q9UGN5 1/20 0.30
PARP4 Q9UKK3 1/20 0.30
PARP3 Q9Y6F1 1/20 0.30
KMT2A Q03164 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
HCRTR2 O43614 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4045088 0.90 CTSS (0.37) CTSKPTGER2CALCRLCTSBCTSS
SCHEMBL4045645 0.88 SMYD3 (0.34) CTSKPTGER2F2CTSBCTSS
SCHEMBL4052140 0.85 HSD17B10 (0.36) CTSKALDH1A1KMT2AHCRTR2
SCHEMBL4048509 0.85 CTSK (0.38) CTSKPAX8F2ALDH1A1SIGMAR1
SCHEMBL4044151 0.84 CTSK (0.43) CTSKCTSSALDH1A1L3MBTL1
SCHEMBL4051458 0.84 CTSK (0.36) CTSKCALCRL
SCHEMBL4050112 0.82 CTSK (0.38) CTSKPAX8F2ALDH1A1SIGMAR1
SCHEMBL4043616 0.80 CTSK (0.35) CTSKPAX8ALDH1A1L3MBTL1
SCHEMBL4044148 0.80 CTSK (0.42) CTSKCTSBCTSS
SCHEMBL4046060 0.79 CTSK (0.35) CTSKPAX8F2ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed