SCHEMBL4053207

SCHEMBL4053207

CCCNCC(O)c1cccnc1

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 11/20 0.57
ADRB2 P07550 7/20 0.57
ADRB3 P13945 17/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25229181 1.00 ADRB1 (0.57) ADRB1ADRB2ADRB3
SCHEMBL30488096 1.00 ADRB1 (0.57) ADRB1ADRB2ADRB3
SCHEMBL30488093 1.00 ADRB1 (0.57) ADRB1ADRB2ADRB3
SCHEMBL30488191 1.00 ADRB1 (0.57) ADRB1ADRB2ADRB3
SCHEMBL25226428 1.00 ADRB1 (0.57) ADRB1ADRB2ADRB3
SCHEMBL20819407 0.91 ADRB1 (0.55) ADRB1ADRB2ADRB3
SCHEMBL26177226 0.84 ADRB3 (0.55) ADRB1ADRB2ADRB3
SCHEMBL11746227 0.84 ADRB1 (0.54) ADRB1ADRB2ADRB3
SCHEMBL6320255 0.80 SLC6A3 (0.55) ADRB1ADRB2ADRB3
SCHEMBL4048311 0.80 SLC6A3 (0.55) ADRB1ADRB2ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250353851-A1 PURINES AND METHODS OF THEIR USE KINETA INC (US) 2025-11-20 US disclosed
EP-4444312-A2 PURINES AND METHODS OF THEIR USE Kineta, Inc. (US) 2024-10-16 EP disclosed
US-20230339890-A1 AMINO ALCOHOL COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. 2023-10-26 US disclosed
US-20230339890-A1 AMINO ALCOHOL COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. 2023-10-26 US disclosed
US-20230339890-A1 AMINO ALCOHOL COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. 2023-10-26 US disclosed
WO-2023107630-A2 AMINO ALCOHOL COMPOUNDS AND USES THEREOF Kineta, Inc. (US) 2023-06-15 WO disclosed
WO-2023107630-A2 AMINO ALCOHOL COMPOUNDS AND USES THEREOF Kineta, Inc. (US) 2023-06-15 WO disclosed
WO-2023107552-A2 PURINES AND METHODS OF THEIR USE Kineta, Inc. (US) 2023-06-15 WO disclosed
WO-2023107552-A2 PURINES AND METHODS OF THEIR USE Kineta, Inc. (US) 2023-06-15 WO disclosed
US-7560474-B2 Derivatives of pyridilethanol (phenylethyl) amines as inhibitors of cholesterol biosynthesis, process for their preparation and pharmaceutical compositions containing them LEK PHARMACEUTICALS D.D. (SI) 2009-07-14 US disclosed
US-20050256172-A1 Novel derivatives of pyridilethanol (phenylethyl) amines as inhibitors of cholesterol biosynthesis, process for their preparation and pharmaceutical compositions containing them LEK PHARMACEUTICALS D.D. (SI) 2005-11-17 US disclosed
CN-1668594-A New derivatives of pyridylethanol (phenylethyl) amines useful as cholesterol biosynthesis inhibitors, process for their preparation and pharmaceutical compositions containing them LEK FARMACEVTSKA DRUZBA DD (SI) 2005-09-14 CN disclosed
EP-1546105-A1 NOVEL DERIVATIVES OF PYRIDYLETHANOL (PHENYLETHYL) AMINES AS INHIBITORS OF CHOLESTEROL BIOSYNTHESIS, PROCESSES FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Lek Pharmaceutical and Chemical Co. D.D. (SI) 2005-06-29 EP disclosed
WO-2004007456-A1 NOVEL DERIVATIVES OF PYRIDYLETHANOL (PHENYLETHYL) AMINES AS INHIBITORS OF CHOLESTEROL BIOSYNTHESIS, PROCESSES FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LEK PHARMACEUTICALS D.D. (SI) 2004-01-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050256172-A1 Novel derivatives of pyridilethanol (phenylethyl) amines as inhibitors of cholesterol biosynthesis, process for their preparation and pharmaceutical compositions containing them DHCR7, NR1H3, NR1H4 ADRB1 35/4885ADRB2 39/4885ADRB3 71/4885
US-20230339890-A1 AMINO ALCOHOL COMPOUNDS AND USES THEREOF AADAT, SLC1A2, SLC1A1 ADRB1 2287/4885ADRB2 2325/4885ADRB3 1624/4885
US-20250353851-A1 PURINES AND METHODS OF THEIR USE TDP1, TDP2, PIKFYVE ADRB1 4582/4885ADRB2 4532/4885ADRB3 4264/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.