SCHEMBL4055280

SCHEMBL4055280

COC(=O)CCC(C#N)(CCC(=O)OC)c1cccc2c1c1cc(OCF)ccc1n2C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
MAPT P10636 2/20 0.34
HPGD P15428 2/20 0.34
TSHR P16473 1/20 0.34
MYLK Q15746 4/20 0.33
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
AS3MT Q9HBK9 3/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
HTT P42858 1/20 0.32
HSD17B10 Q99714 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
GABRA1 P14867 1/20 0.32
GABRG2 P18507 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4375180 0.76 PSEN1 (0.38) ALDH1A1KDM4EMAPTHPGDTSHR
SCHEMBL4055284 0.72 CASP3 (0.36) ALDH1A1KDM4EMAPTHPGDKMT2A
SCHEMBL4052668 0.69 MAPT (0.43) ALDH1A1KDM4EMAPTHPGDMYLK
SCHEMBL11821422 0.68 CYP1A2 (0.48) ALDH1A1KDM4EMAPTHPGDTSHR
SCHEMBL11920949 0.67 ALDH1A1 (0.39) ALDH1A1KDM4EMAPTHPGDTSHR
SCHEMBL4053047 0.67 ALDH1A1 (0.39) ALDH1A1MAPTMEN1KMT2ANPC1
SCHEMBL8021561 0.66 ALDH1A1 (0.39) ALDH1A1KDM4EMAPTHPGDTSHR
SCHEMBL4239306 0.66 POLB (0.34) ALDH1A1KDM4EMAPTHPGDTSHR
SCHEMBL4373655 0.65 MEN1 (0.66) ALDH1A1KDM4EMAPTHPGDTSHR
SCHEMBL11093234 0.65 ALDH1A1 (0.39) ALDH1A1KDM4EMAPTHPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO disclosed