SCHEMBL4055284

SCHEMBL4055284

COC(=O)CCC(C#N)(CCC(=O)OC)c1ccc(OC)c2c1c1cc(F)ccc1n2C

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.36
KDM4E B2RXH2 4/20 0.35
PLA2G4A P47712 1/20 0.33
ALDH1A1 P00352 4/20 0.33
HPGD P15428 2/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
HK1 P19367 1/20 0.33
HKDC1 Q2TB90 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CNR1 P21554 3/20 0.33
AVPR1B P47901 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
TP53 P04637 1/20 0.31
KMT2A Q03164 1/20 0.31
ATM Q13315 1/20 0.31
AR P10275 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4053047 0.87 ALDH1A1 (0.39) PLA2G4AALDH1A1MAPTNPSR1TP53
SCHEMBL4375183 0.75 KDM4E (0.37) CASP3KDM4EPLA2G4AALDH1A1LMNA
SCHEMBL4055280 0.72 ALDH1A1 (0.35) KDM4EALDH1A1HPGDMAPTHSD17B10
SCHEMBL4053668 0.71 KDM4E (0.39) KDM4EPLA2G4AALDH1A1HPGDLMNA
SCHEMBL11822888 0.70 HSD17B10 (0.46) KDM4EALDH1A1HPGDLMNAMAPT
SCHEMBL6623387 0.69 KDM4E (0.44) KDM4EALDH1A1HPGDLMNAMAPT
SCHEMBL4052669 0.69 KDM4E (0.41) KDM4EPLA2G4AALDH1A1HPGDHSD17B10
SCHEMBL11821360 0.68 CA12 (0.41) KDM4EALDH1A1HPGDLMNAMAPT
SCHEMBL11825374 0.68 MAPT (0.37) KDM4EALDH1A1HPGDLMNAMAPT
SCHEMBL7375552 0.68 HSD17B10 (0.64) ALDH1A1MAPTHSD17B10CNR1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO disclosed